Robust Synthesis of Tetra-Boronate Esters Analogues and the Corresponding Boronic Acids Derivatives
學年 110
學期 2
出版（發表）日期 2022-05-02
作品名稱 Robust Synthesis of Tetra-Boronate Esters Analogues and the Corresponding Boronic Acids Derivatives
作品名稱（其他語言）
著者 Shuo-Bei Qiu, Jing-Han Xiao, Pin-Rui Chen, Guan-Lin Ai, Kuan-Lin Pan, Jen-Kun Chen, Yi-Wei Chen, and Po-Shen Pan
單位
出版者
著錄名稱、卷期、頁數 European Journal of Organic Chemistry 2022(31),　e202200379
摘要 Organoboron compounds are widely used in catalytic reactions, medicinal chemistry, chemosensors, and polymer applications, because of their low toxicity, high stability, Lewis acidity, chemical versatility, and ability to form covalent bonds with their nucleophilic targets, In this report, we demonstrate how to efficiently assemble tetra boronate-containing compounds at the gram-scale via a one-pot modified microwave-assisted Ugi-4CR reaction. These boronate esters can then be transformed into the corresponding boronic acids under a reliable deprotection method, also reported herein.
關鍵字 Boronic acid; Deprotection; Microwave chemistry; Multicomponent reactions; Ugi-4CR
語言 zh_TW
ISSN 1099-0690
期刊性質 國外
收錄於 SCI
產學合作
通訊作者 Po-Shen Pan
審稿制度 是
國別 DEU
公開徵稿
出版型式 ,電子版,紙本
相關連結

機構典藏連結 ( http://tkuir.lib.tku.edu.tw:8080/dspace/handle/987654321/124323 )