標題:Synthesis of boron-containing tetrazoles under neutral microwave-assisted conditions |
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學年 | 108 |
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學期 | 1 |
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出版(發表)日期 | 2019/10/01 |
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作品名稱 | Synthesis of boron-containing tetrazoles under neutral microwave-assisted conditions |
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作品名稱(其他語言) | |
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著者 | Yu-Yun Chen; Wan-Xin Lin; Kai-Wei Hsu; Wan-Chi Li; Chih-Hsuan Wang; Jui-Ping Yu; Chia-Wen Chang; Shuo-Bei Qiu; Po-Shiuan Hsieh; Yi-Wei Chen; Po-Shen Pan |
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單位 | |
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出版者 | |
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著錄名稱、卷期、頁數 | Research on Chemical Intermediates 45, p.5375–5388 |
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摘要 | In this report, the mild synthetic strategies for the synthesis of two series of boron-containing tetrazoles were included. For the first series, a boron-containing isocyanide reacted with TMS-N3 to afford the desire products. The reaction took place at 60 °C in TFE for 30 min under microwave irradiation. For the second series, the Ugi four-component reaction (Ugi-4CR) was deployed to synthesize the desire products. The reaction took place simply in MeOH at ambient temperature for 2 h. The synthetic strategies included could provide access to ranges of boron-containing tetrazole libraries, which might possess unique biological properties. |
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關鍵字 | Boron;Tetrazoles;Ugi;Microwave;Multicomponent reaction;Boron neutron capture therapy |
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語言 | 英文(美國) |
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ISSN | 1568-5675 |
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期刊性質 | 國外 |
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收錄於 | SCI; |
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產學合作 | |
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通訊作者 | Po-Shen Pan |
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審稿制度 | 否 |
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國別 | 德國 |
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公開徵稿 | |
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出版型式 | ,電子版 |
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