Synthesis of boron-containing tetrazoles under neutral microwave-assisted conditions
學年 108
學期 1
出版（發表）日期 2019-10-01
作品名稱 Synthesis of boron-containing tetrazoles under neutral microwave-assisted conditions
作品名稱（其他語言）
著者 Yu-Yun Chen; Wan-Xin Lin; Kai-Wei Hsu; Wan-Chi Li; Chih-Hsuan Wang; Jui-Ping Yu; Chia-Wen Chang; Shuo-Bei Qiu; Po-Shiuan Hsieh; Yi-Wei Chen; Po-Shen Pan
單位
出版者
著錄名稱、卷期、頁數 Research on Chemical Intermediates 45, p.5375–5388
摘要 In this report, the mild synthetic strategies for the synthesis of two series of boron-containing tetrazoles were included. For the first series, a boron-containing isocyanide reacted with TMS-N3 to afford the desire products. The reaction took place at 60 °C in TFE for 30 min under microwave irradiation. For the second series, the Ugi four-component reaction (Ugi-4CR) was deployed to synthesize the desire products. The reaction took place simply in MeOH at ambient temperature for 2 h. The synthetic strategies included could provide access to ranges of boron-containing tetrazole libraries, which might possess unique biological properties.
關鍵字 Boron;Tetrazoles;Ugi;Microwave;Multicomponent reaction;Boron neutron capture therapy
語言 en_US
ISSN 1568-5675
期刊性質 國外
收錄於 SCI
產學合作
通訊作者 Po-Shen Pan
審稿制度 否
國別 DEU
公開徵稿
出版型式 ,電子版
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